6 minute read
Mar. 26, 2024

Lirafugratinib (RLY-4008): The First Isoform-Selective FGFR2 Inhibitor with Potential Best-in-Class Properties

lirafugratinib (RLY-4008)

oral covalent FGFR2 inhibitor Ph. II for cholangiocarcinoma from rational design with MD simulations Cancer Discov., June 4, 2023 Relay Therapeutics, MA / D. E. Shaw Research, NY

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